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MM 11253
CAS No. 345952-44-5
MM 11253( MM-11253 )
Catalog No. M27662 CAS No. 345952-44-5
MM 11253 is a RARγ antagonist with IC50 of 44nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 72 | Get Quote |
|
| 10MG | 115 | Get Quote |
|
| 25MG | 260 | Get Quote |
|
| 50MG | 410 | Get Quote |
|
| 100MG | 605 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameMM 11253
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NoteResearch use only, not for human use.
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Brief DescriptionMM 11253 is a RARγ antagonist with IC50 of 44nM.
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DescriptionMM 11253 is a RARγ antagonist with IC50 of 44nM.(In Vitro):MM11253 blocks the ability of MM11254 and MM11389 to inhibit squamous cell carcinoma cell growth .
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In VitroMM11253 blocks the ability of MM11254 and MM11389 to inhibit squamous cell carcinoma cell growth.
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In Vivo——
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SynonymsMM-11253
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PathwayMetabolic Enzyme/Protease
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TargetRetinoid Receptor
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RecptorAMPK α2β2γ1|AMPK α1β1γ1|AMPK α2β1γ1|AMPK α1β2γ1
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Research Area——
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Indication——
Chemical Information
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CAS Number345952-44-5
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Formula Weight462.67
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Molecular FormulaC28H30O2S2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (270.17 mM)
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SMILESCC1(C)CCC(C)(C)c2cc(ccc12)C1(SCCS1)c1ccc2cc(ccc2c1)C(O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Zhang LN, et al. Novel small-molecule AMP-activated protein kinase allosteric activator with beneficial effects in db/db mice. PLoS One. 2013 Aug 20;8(8):e72092.
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